Orphan GPCRs


Human	GPR4 G protein-coupled receptor 4
Human	GPR65 G protein-coupled receptor 65
Human	GPR68 G protein-coupled receptor 68
Human	GPR132 G protein-coupled receptor 132
Human	P2RY8 P2Y receptor family member 8
Human	AGTR2 angiotensin ⅠⅠ receptor type 2
Human	GPRC6A G protein-coupled receptor class C group 6 member A
Human	CCRL2 C-C motif chemokine receptor like 2
Human	ACKR3 atypical chemokine receptor 3
Human	GPR1 G protein-coupled receptor 1
Human	GPR3 G protein-coupled receptor 3
Human	GPR6 G protein-coupled receptor 6
Human	GPR12 G protein-coupled receptor 12
Human	GPR15 G protein-coupled receptor 15
Human	GPR17 G protein-coupled receptor 17
Human	GPR18 G protein-coupled receptor 18
Human	GPR19 G protein-coupled receptor 19
Human	GPR20 G protein-coupled receptor 20
Human	GPR21 G protein-coupled receptor 21
Human	GPR22 G protein-coupled receptor 22
Human	GPR25 G protein-coupled receptor 25
Human	GPR26 G protein-coupled receptor 26
Human	GPR27 G protein-coupled receptor 27
Human	GPR31 G protein-coupled receptor 31
Human	GPR32 G protein-coupled receptor 32
Human	GPR35 G protein-coupled receptor 35
Human	GPR37 G protein-coupled receptor 37
Human	GPR37L1 G protein-coupled receptor 37 like 1
Human	GPR39 G protein-coupled receptor 39
Human	GPR45 G protein-coupled receptor 45
Human	GPR50 G protein-coupled receptor 50
Human	GPR52 G protein-coupled receptor 52
Human	GPR61 G protein-coupled receptor 61
Human	GPR62 G protein-coupled receptor 62
Human	GPR63 G protein-coupled receptor 63
Human	GPR75 G protein-coupled receptor 75
Human	GPR78 G protein-coupled receptor 78
Human	GPR82 G protein-coupled receptor 82
Human	GPR83 G protein-coupled receptor 83
Human	GPR85 G protein-coupled receptor 85
Human	GPR87 G protein-coupled receptor 87
Human	GPR88 G protein-coupled receptor 88
Human	GPR101 G protein-coupled receptor 101
Human	GPR135 G protein-coupled receptor 135
Human	GPR139 G protein-coupled receptor 139
Human	GPR141 G protein-coupled receptor 141
Human	GPR142 G protein-coupled receptor 142
Human	GPR146 G protein-coupled receptor 146
Human	GPR148 G protein-coupled receptor 148
Human	GPR149 G protein-coupled receptor 149

12…4

Species	Receptor	Family	Assays
Mouse	Ackr3 atypical chemokine receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr1 G protein-coupled receptor 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr3 G-protein coupled receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr6 G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr12 G-protein coupled receptor 12	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr17 G protein-coupled receptor 17	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr18 G protein-coupled receptor 18	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr19 G protein-coupled receptor 19	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr20 G protein-coupled receptor 20	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr21 G protein-coupled receptor 21	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr22 G protein-coupled receptor 22	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr25 G protein-coupled receptor 25	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr26 G protein-coupled receptor 26	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr27 G protein-coupled receptor 27	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr35 G protein-coupled receptor 35	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: zaprinast EC50: 700 nM
Mouse	Gpr37 G protein-coupled receptor 37	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr37l1 G protein-coupled receptor 37-like 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr39 G protein-coupled receptor 39	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr45 G protein-coupled receptor 45	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr61 G protein-coupled receptor 61	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr63 G protein-coupled receptor 63	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr75 G protein-coupled receptor 75	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr82 G protein-coupled receptor 82	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr83 G protein-coupled receptor 83	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr85 G protein-coupled receptor 85	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr87 G protein-coupled receptor 87	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr88 G-protein coupled receptor 88	Orphan GPCRs	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr135 G protein-coupled receptor 135	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr146 G protein-coupled receptor 146	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr150 G protein-coupled receptor 150	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr151 G protein-coupled receptor 151	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr152 G protein-coupled receptor 152	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr160 G protein-coupled receptor 160	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr162 G protein-coupled receptor 162	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr171 G protein-coupled receptor 171	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr173 G-protein coupled receptor 173	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr182 G protein-coupled receptor 182	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Lgr6 leucine-rich repeat-containing G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mas1 MAS1 oncogene	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprd MAS-related GPR, member D	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgpre MAS-related GPR, member E	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprf MAS-related GPR, member F	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprg MAS-related GPR, member G	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprx1 MAS-related GPR, member X1	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar2 trace amine-associated receptor 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar5 trace amine-associated receptor 5	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar6 trace amine-associated receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar8a trace amine-associated receptor 8A	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar9 trace amine-associated receptor 9	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr157 G protein-coupled receptor 157	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:

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