Orphan GPCRs


Human	GPR150 G protein-coupled receptor 150
Human	GPR151 G protein-coupled receptor 151
Human	GPR152 G protein-coupled receptor 152
Human	GPR153 G protein-coupled receptor 153
Human	GPR160 G protein-coupled receptor 160
Human	GPR161 G protein-coupled receptor 161
Human	GPR162 G protein-coupled receptor 162
Human	GPR171 G protein-coupled receptor 171
Human	GPR173 G protein-coupled receptor 173
Human	GPR182 G protein-coupled receptor 182
Human	LGR4 leucine rich repeat containing G protein-coupled receptor 4
Human	LGR5 leucine rich repeat containing G protein-coupled receptor 5
Human	LGR6 leucine rich repeat containing G protein-coupled receptor 6
Human	MAS1 MAS1 proto-oncogene, G protein-coupled receptor
Human	MAS1L MAS1 proto-oncogene like, G protein-coupled receptor
Human	MRGPRD MAS related GPR family member D
Human	MRGPRE MAS related GPR family member E
Human	MRGPRF MAS related GPR family member F
Human	MRGPRG MAS related GPR family member G
Human	MRGPRX1 MAS related GPR family member X1
Human	MRGPRX2 MAS related GPR family member X2
Human	MRGPRX3 MAS related GPR family member X3
Human	MRGPRX4 MAS related GPR family member X4
Human	TAAR2 trace amine associated receptor 2
Human	TAAR5 trace amine associated receptor 5
Human	TAAR6 trace amine associated receptor 6
Human	TAAR8 trace amine associated receptor 8
Human	TAAR9 trace amine associated receptor 9
Human	GPR143 G protein-coupled receptor 143
Human	GPR157 G protein-coupled receptor 157
Human	GPR156 G protein-coupled receptor 156
Human	GPR158 G protein-coupled receptor 158
Human	GPER1 G protein-coupled estrogen receptor 1
Human	GPRC5A G protein-coupled receptor class C group 5 member A
Human	GPRC5B G protein-coupled receptor class C group 5 member B
Human	GPRC5C G protein-coupled receptor class C group 5 member C
Human	GPRC5D G protein-coupled receptor class C group 5 member D
Human	ACKR2 atypical chemokine receptor 2
Human	ACKR4 atypical chemokine receptor 4
Human	ACKR1 atypical chemokine receptor 1 (Duffy blood group)
Human	GPR176 G protein-coupled receptor 176
Human	GPR107 G protein-coupled receptor 107
Human	GPR137 G protein-coupled receptor 137
Human	TPRA1 transmembrane protein adipocyte associated 1
Mouse	Gpr4 G protein-coupled receptor 4
Mouse	Gpr65 G-protein coupled receptor 65
Mouse	Gpr68 G protein-coupled receptor 68
Mouse	Gpr132 G protein-coupled receptor 132
Mouse	Agtr2 angiotensin ⅠⅠ receptor, type 2
Mouse	Ccrl2 chemokine (C-C motif) receptor-like 2

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Species	Receptor	Family	Assays
Mouse	Ackr3 atypical chemokine receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr1 G protein-coupled receptor 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr3 G-protein coupled receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr6 G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr12 G-protein coupled receptor 12	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr17 G protein-coupled receptor 17	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr18 G protein-coupled receptor 18	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr19 G protein-coupled receptor 19	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr20 G protein-coupled receptor 20	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr21 G protein-coupled receptor 21	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr22 G protein-coupled receptor 22	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr25 G protein-coupled receptor 25	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr26 G protein-coupled receptor 26	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr27 G protein-coupled receptor 27	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr35 G protein-coupled receptor 35	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: zaprinast EC50: 700 nM
Mouse	Gpr37 G protein-coupled receptor 37	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr37l1 G protein-coupled receptor 37-like 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr39 G protein-coupled receptor 39	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr45 G protein-coupled receptor 45	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr61 G protein-coupled receptor 61	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr63 G protein-coupled receptor 63	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr75 G protein-coupled receptor 75	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr82 G protein-coupled receptor 82	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr83 G protein-coupled receptor 83	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr85 G protein-coupled receptor 85	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr87 G protein-coupled receptor 87	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr88 G-protein coupled receptor 88	Orphan GPCRs	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr135 G protein-coupled receptor 135	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr146 G protein-coupled receptor 146	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr150 G protein-coupled receptor 150	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr151 G protein-coupled receptor 151	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr152 G protein-coupled receptor 152	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr160 G protein-coupled receptor 160	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr162 G protein-coupled receptor 162	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr171 G protein-coupled receptor 171	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr173 G-protein coupled receptor 173	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr182 G protein-coupled receptor 182	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Lgr6 leucine-rich repeat-containing G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mas1 MAS1 oncogene	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprd MAS-related GPR, member D	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgpre MAS-related GPR, member E	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprf MAS-related GPR, member F	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprg MAS-related GPR, member G	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Mrgprx1 MAS-related GPR, member X1	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar2 trace amine-associated receptor 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar5 trace amine-associated receptor 5	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar6 trace amine-associated receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar8a trace amine-associated receptor 8A	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Taar9 trace amine-associated receptor 9	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Mouse	Gpr157 G protein-coupled receptor 157	Orphan GPCRs	Available Assay modes: Agonist Panels: Mouse orphan GPCRs ⋅ à la carte	Reference agonist: EC50:

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