Human BRS3

Figure. Concentration-dependent activation of BRS3 by bombesin

Reporter cells were transfected with either the expression plasmid for human bombesin receptor subtype 3 (BRS3) or the mock plasmid and treated with various concentrations of bombesin. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 2.4 nM.

Nomenclature
bombesin receptor subtype 3
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Immunology/Infection, Oncology, Hematology, Endocrinology/Metabolism, Ophthalmology, Respiratory, Dermatology, Urology/Reproduction, Human non-orphan GPCRs

BRS3 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors