Human GIPR

Figure. Concentration-dependent activation of GIPR by GIP

Reporter cells were transfected with either the expression plasmid for human gastric inhibitory polypeptide receptor (GIPR) or the mock plasmid and treated with various concentrations of GIP. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 3.4 nM.

Nomenclature
gastric inhibitory polypeptide receptor
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Endocrinology/Metabolism, Human non-orphan GPCRs

GIPR orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors

Filters Sort results
Reset Apply