Human KISS1R

Figure. Concentration-dependent activation of KISS1R by kisspeptin‐10

Reporter cells were transfected with either the expression plasmid for human KISS1 receptor (KISS1R) or the mock plasmid and treated with various concentrations of kisspeptin‐10. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 1.3 nM.

Nomenclature
KISS1 receptor
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Oncology, Endocrinology/Metabolism, Neurology, Ophthalmology, Gastrointestinal, Dermatology, Musculoskeletal, Urology/Reproduction, Human non-orphan GPCRs

KISS1R orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors

Filters Sort results
Reset Apply