Human NTSR1

Figure. Concentration-dependent activation of NTSR1 by neurotensin

Reporter cells were transfected with either the expression plasmid for human neurotensin receptor 1 (NTSR1) or the mock plasmid and treated with various concentrations of neurotensin. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 180 pM.

Nomenclature
neurotensin receptor 1
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Oncology, Psychiatry, Human non-orphan GPCRs

NTSR1 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors