Human GPR88

Figure. Concentration-dependent activation of GPR88 by 2‐PCCA

Reporter cells were transfected with the expression plasmid for human G protein-coupled receptor 88 (GPR88) and treated with various concentrations of 2‐PCCA. Data points shown are the mean ± SEM of an experiment (n = 4), and the curve is a fit to Hill equation with an EC50 of 1.0 µM.

Nomenclature
G protein-coupled receptor 88
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Human orphan GPCRs

GPR88 orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors

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