Human PTAFR

Figure. Concentration-dependent activation of PTAFR by CH3‐carbamyl PAF C‐16

Reporter cells were transfected with either the expression plasmid for human platelet activating factor receptor (PTAFR) or the mock plasmid and treated with various concentrations of CH3‐carbamyl PAF C‐16. Data points shown are the mean ± SEM of an experiment (n = 3), and the curve is a fit to Hill equation with an EC50 of 840 pM.

Nomenclature
platelet activating factor receptor
Available assay modes
Agonist, Inverse agonist, Antagonist, PAM, NAM
Panels
à la carte, Immunology/Infection, Hematology, Ophthalmology, Cardiology, Respiratory, Gastrointestinal, Urology/Reproduction, Human non-orphan GPCRs

PTAFR orthologs in other animal species including rat, rabbit, dog, and macaque monkey are ready upon request.

Related Receptors