Adrenoceptors


Human	ADRA1A adrenoceptor alpha 1A
Human	ADRA1B adrenoceptor alpha 1B
Human	ADRA1D adrenoceptor alpha 1D
Human	ADRA2A adrenoceptor alpha 2A
Human	ADRA2B adrenoceptor alpha 2B
Human	ADRA2C adrenoceptor alpha 2C
Human	ADRB1 adrenoceptor beta 1
Human	ADRB2 adrenoceptor beta 2
Human	ADRB3 adrenoceptor beta 3
Mouse	Adra1a adrenergic receptor, alpha 1a
Mouse	Adra1b adrenergic receptor, alpha 1b
Mouse	Adra1d adrenergic receptor, alpha 1d
Mouse	Adra2a adrenergic receptor, alpha 2a
Mouse	Adra2b adrenergic receptor, alpha 2b
Mouse	Adra2c adrenergic receptor, alpha 2c
Mouse	Adrb1 adrenergic receptor, beta 1
Mouse	Adrb2 adrenergic receptor, beta 2
Mouse	Adrb3 adrenergic receptor, beta 3

Species	Receptor	Family	Assays
Human	ADRA1A adrenoceptor alpha 1A	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety ⋅ Safety Premium ⋅ Immunology/Infection ⋅ Oncology ⋅ Hematology ⋅ Endocrinology/Metabolism ⋅ Ophthalmology ⋅ Cardiology ⋅ Respiratory ⋅ Gastrointestinal ⋅ Dermatology ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: L‐phenylephrine EC50: 18 nM
Human	ADRA1B adrenoceptor alpha 1B	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety Premium ⋅ Neurology ⋅ Cardiology ⋅ à la carte	Reference agonist: L‐phenylephrine EC50: 28 nM
Human	ADRA1D adrenoceptor alpha 1D	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety Premium ⋅ à la carte	Reference agonist: L‐phenylephrine EC50: 67 nM
Human	ADRA2A adrenoceptor alpha 2A	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety ⋅ Safety Premium ⋅ Psychiatry ⋅ Cardiology ⋅ Dermatology ⋅ Musculoskeletal ⋅ à la carte	Reference agonist: noradrenaline EC50: 71 nM
Human	ADRA2B adrenoceptor alpha 2B	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety Premium ⋅ Immunology/Infection ⋅ Oncology ⋅ Hematology ⋅ Psychiatry ⋅ Neurology ⋅ Ophthalmology ⋅ Cardiology ⋅ Respiratory ⋅ Gastrointestinal ⋅ Dermatology ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: noradrenaline EC50: 33 nM
Human	ADRA2C adrenoceptor alpha 2C	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety Premium ⋅ Cardiology ⋅ à la carte	Reference agonist: noradrenaline EC50: 89 nM
Human	ADRB1 adrenoceptor beta 1	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety ⋅ Safety Premium ⋅ Endocrinology/Metabolism ⋅ Psychiatry ⋅ Cardiology ⋅ Gastrointestinal ⋅ à la carte	Reference agonist: isoproterenol EC50: 22 nM
Human	ADRB2 adrenoceptor beta 2	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety ⋅ Safety Premium ⋅ Immunology/Infection ⋅ Oncology ⋅ Hematology ⋅ Endocrinology/Metabolism ⋅ Psychiatry ⋅ Neurology ⋅ Ophthalmology ⋅ Cardiology ⋅ Respiratory ⋅ Gastrointestinal ⋅ Dermatology ⋅ Musculoskeletal ⋅ Urology/Reproduction ⋅ à la carte	Reference agonist: isoproterenol EC50: 26 nM
Human	ADRB3 adrenoceptor beta 3	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human non-orphan GPCRs ⋅ Safety Premium ⋅ Endocrinology/Metabolism ⋅ Cardiology ⋅ à la carte	Reference agonist: isoproterenol EC50: 47 nM
Mouse	Adra1a adrenergic receptor, alpha 1a	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: L‐phenylephrine EC50: 73 nM
Mouse	Adra1b adrenergic receptor, alpha 1b	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: L‐phenylephrine EC50: 82 nM
Mouse	Adra1d adrenergic receptor, alpha 1d	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: L‐phenylephrine EC50: 77 nM
Mouse	Adra2a adrenergic receptor, alpha 2a	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: noradrenaline EC50: 480 nM
Mouse	Adra2b adrenergic receptor, alpha 2b	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: noradrenaline EC50: 110 nM
Mouse	Adra2c adrenergic receptor, alpha 2c	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: noradrenaline EC50: 250 nM
Mouse	Adrb1 adrenergic receptor, beta 1	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: isoproterenol EC50: 32 nM
Mouse	Adrb2 adrenergic receptor, beta 2	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: isoproterenol EC50: 59 nM
Mouse	Adrb3 adrenergic receptor, beta 3	Adrenoceptors	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Mouse non-orphan GPCRs ⋅ à la carte	Reference agonist: isoproterenol EC50: 97 nM