Orphan GPCRs


Mouse	Gper1 G protein-coupled estrogen receptor 1
Mouse	Gprc5c G protein-coupled receptor, family C, group 5, member C
Mouse	Ackr2 atypical chemokine receptor 2
Mouse	Ackr4 atypical chemokine receptor 4
Mouse	Ackr1 atypical chemokine receptor 1 (Duffy blood group)
Mouse	Gpr107 G protein-coupled receptor 107
Mouse	Tpra1 transmembrane protein, adipocyte asscociated 1

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Species	Receptor	Family	Assays
Human	GPR4 G protein-coupled receptor 4	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR65 G protein-coupled receptor 65	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR68 G protein-coupled receptor 68	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR132 G protein-coupled receptor 132	Orphan GPCRs ⋅	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	P2RY8 P2Y receptor family member 8	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	AGTR2 angiotensin ⅠⅠ receptor type 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPRC6A G protein-coupled receptor class C group 6 member A	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	CCRL2 C-C motif chemokine receptor like 2	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	ACKR3 atypical chemokine receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR1 G protein-coupled receptor 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR3 G protein-coupled receptor 3	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR6 G protein-coupled receptor 6	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR12 G protein-coupled receptor 12	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR15 G protein-coupled receptor 15	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR17 G protein-coupled receptor 17	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR18 G protein-coupled receptor 18	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR19 G protein-coupled receptor 19	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR20 G protein-coupled receptor 20	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR21 G protein-coupled receptor 21	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR22 G protein-coupled receptor 22	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR25 G protein-coupled receptor 25	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR26 G protein-coupled receptor 26	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR27 G protein-coupled receptor 27	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR31 G protein-coupled receptor 31	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR32 G protein-coupled receptor 32	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR35 G protein-coupled receptor 35	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: zaprinast EC50: 2.8 µM
Human	GPR37 G protein-coupled receptor 37	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR37L1 G protein-coupled receptor 37 like 1	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR39 G protein-coupled receptor 39	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR45 G protein-coupled receptor 45	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR50 G protein-coupled receptor 50	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR52 G protein-coupled receptor 52	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR61 G protein-coupled receptor 61	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR62 G protein-coupled receptor 62	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR63 G protein-coupled receptor 63	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR75 G protein-coupled receptor 75	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR78 G protein-coupled receptor 78	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR82 G protein-coupled receptor 82	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR83 G protein-coupled receptor 83	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR85 G protein-coupled receptor 85	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR87 G protein-coupled receptor 87	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR88 G protein-coupled receptor 88	Orphan GPCRs	Available Assay modes: Agonist ⋅ Inverse agonist ⋅ Antagonist ⋅ PAM ⋅ NAM Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: 2‐PCCA EC50: 1.0 µM
Human	GPR101 G protein-coupled receptor 101	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR135 G protein-coupled receptor 135	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR139 G protein-coupled receptor 139	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR141 G protein-coupled receptor 141	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR142 G protein-coupled receptor 142	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR146 G protein-coupled receptor 146	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR148 G protein-coupled receptor 148	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:
Human	GPR149 G protein-coupled receptor 149	Orphan GPCRs	Available Assay modes: Agonist Panels: Human orphan GPCRs ⋅ à la carte	Reference agonist: EC50:

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